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Target Name *
Alternative Names
UniProt ID
(optional)
Effect Type
(pick 1–3)
brain
sleep
pain
cardiovascular
immune
gut
diabetes
weight loss
reproductive
muscle
skin
inflammation
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00
all
64
01
BRAIN
15
02
SLEEP
1
03
PAIN
7
04
CARDIOVASCULAR
9
05
IMMUNE
1
06
GUT
9
07
DIABETES
4
08
WEIGHT LOSS
10
09
REPRODUCTIVE
6
10
MUSCLE
9
11
SKIN
4
12
INFLAMMATION
9
13
CANCER
3
14
AGING
13
64 targets
·
sorted by activity
activity
a-z
502
cards
ACE
angiotensin-converting enzyme
metalloprotease
+ CARDIOVASCULAR
CALCR/RAMP
PTH1R
+6
300
cards
Antimicrobial
category
AMP
+ IMMUNE · INFLAMMATION
VPAC1
TACR1
+6
228
cards
GLP-1R
GLP-1 receptor
secretin receptor family (class B GPCR)
+ WEIGHT LOSS · DIABETES · GUT
NTSR1
CCKAR
+14
199
cards
Anticancer
category
+ CANCER
GNRHR
IGF-1R
33
cards
OPRM1
mu-opioid receptor
rhodopsin-like GPCR (class A)
+ PAIN
CALCR/RAMP
TACR1
+4
best
4
31
cards
CALCR/RAMP
calcitonin receptor
secretin receptor family (class B GPCR)
+ PAIN · CARDIOVASCULAR
ACE
OPRM1
+12
29
cards
NTSR1
neurotensin-1 receptor
rhodopsin-like GPCR (class A)
+ BRAIN · GUT
GLP-1R
CCKAR
+17
26
cards
CCKAR
CCK1 receptor
rhodopsin-like GPCR (class A)
+ GUT · WEIGHT LOSS
GLP-1R
NTSR1
+13
26
cards
VPAC1
VIP receptor 1
secretin receptor family (class B GPCR)
+ BRAIN · INFLAMMATION · GUT
ANTIMICROBIAL
GLP-1R
+22
25
cards
PTH1R
PTH receptor type 1
secretin-like GPCR (class B)
+ CARDIOVASCULAR · AGING
ACE
CALCR/RAMP
+18
23
cards
GCGR
glucagon receptor
secretin receptor family (class B GPCR)
+ WEIGHT LOSS · DIABETES
GLP-1R
CCKAR
+8
22
cards
MC3R
melanocortin-3 receptor
rhodopsin-like GPCR (class A)
+ WEIGHT LOSS · BRAIN
GLP-1R
NTSR1
+18
20
cards
GHSR
ghrelin receptor
rhodopsin-like GPCR (class A)
+ MUSCLE · GUT · SLEEP
GLP-1R
NTSR1
+14
19
cards
EDNRA
ETA receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE
CALCR/RAMP
+6
19
cards
TACR1
NK1 receptor
rhodopsin-like GPCR (class A)
+ PAIN · BRAIN · INFLAMMATION
ANTIMICROBIAL
OPRM1
+20
18
cards
OPRD1
delta-opioid receptor
rhodopsin-like GPCR (class A)
+ PAIN · BRAIN
OPRM1
CALCR/RAMP
+15
17
cards
GALR1
galanin-1 receptor
rhodopsin-like GPCR (class A)
+ BRAIN · GUT · WEIGHT LOSS
GLP-1R
NTSR1
+21
17
cards
MC2R
melanocortin-2 receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE
CALCR/RAMP
+6
17
cards
MC4R
melanocortin-4 receptor
rhodopsin-like GPCR (class A)
+ WEIGHT LOSS · REPRODUCTIVE · BRAIN
GLP-1R
NTSR1
+21
16
cards
CRHR2
CRF2 receptor
secretin-like GPCR (class B)
+ BRAIN · WEIGHT LOSS
GLP-1R
NTSR1
+18
14
cards
GIPR
GIP receptor
secretin receptor family (class B GPCR)
+ WEIGHT LOSS · DIABETES
GLP-1R
CCKAR
+8
13
cards
ADCYAP1R1 / PAC1R
PAC1 receptor
secretin-like GPCR (class B)
+ PAIN · BRAIN · INFLAMMATION
ANTIMICROBIAL
OPRM1
+20
12
cards
GnRHR
GnRH receptor
rhodopsin-like (class A GPCR)
+ CANCER · REPRODUCTIVE
ANTICANCER
MC4R
+5
12
cards
NPBWR1
neuropeptide B receptor 1
rhodopsin-like GPCR (class A)
+ BRAIN · PAIN
OPRM1
CALCR/RAMP
+15
11
cards
GLP-2R
glucagon-like peptide 2 receptor
secretin-like GPCR (class B)
+ GUT
GLP-1R
NTSR1
+6
10
cards
TACR2
NK2 receptor
rhodopsin-like GPCR (class A)
+ PAIN · GUT · INFLAMMATION
ANTIMICROBIAL
GLP-1R
+17
8
cards
KISS1R
kisspeptin receptor
rhodopsin-like GPCR (class A)
+ REPRODUCTIVE · BRAIN
NTSR1
VPAC1
+15
8
cards
Neuroprotective
category
nootropic
+ BRAIN
NTSR1
VPAC1
+12
8
cards
OXTR
oxytocin receptor
rhodopsin-like GPCR (class A)
+ BRAIN · REPRODUCTIVE
NTSR1
VPAC1
+15
7
cards
AVPR1A
V1a receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE
CALCR/RAMP
+6
7
cards
IGF-1R
insulin-like growth factor 1 receptor
receptor tyrosine kinase
+ MUSCLE · CANCER · AGING
ANTICANCER
PTH1R
+14
7
cards
Longevity
category
+ AGING
PTH1R
IGF-1R
+10
6
cards
AVPR2
vasopressin V2 receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE
CALCR/RAMP
+6
6
cards
Cosmeceutical
category
+ SKIN
MC1R
SKIN PEPTIDES
+1
6
cards
SCTR
secretin receptor
secretin-like GPCR (class B)
+ GUT · BRAIN
GLP-1R
NTSR1
+17
5
cards
AVPR1B
V1b receptor
rhodopsin-like GPCR (class A)
+ BRAIN
NTSR1
VPAC1
+12
5
cards
LHCGR
LH receptor
glycoprotein hormone receptor (class A GPCR)
+ REPRODUCTIVE
MC4R
GNRHR
+3
5
cards
Tissue Repair
category
wound healing
+ INFLAMMATION · AGING
ANTIMICROBIAL
VPAC1
+17
4
cards
MC1R
melanocortin-1 receptor
rhodopsin-like GPCR (class A)
+ SKIN · INFLAMMATION
ANTIMICROBIAL
VPAC1
+9
3
cards
Activin A
INHBA
TGF-β superfamily
+ MUSCLE · AGING · INFLAMMATION
ANTIMICROBIAL
VPAC1
+19
3
cards
GDF-8
myostatin
TGF-β superfamily
+ MUSCLE · WEIGHT LOSS · AGING
GLP-1R
CCKAR
+21
best
0.742
3
cards
GHRHR
Class B GPCR / secretin receptor family
3
cards
Immune
category
3
cards
INSR
insulin receptor
receptor tyrosine kinase
+ DIABETES · AGING
GLP-1R
PTH1R
+13
3
cards
Skin Peptides
category
cosmeceutical
+ SKIN
COSMECEUTICAL
MC1R
+1
2
cards
ActRIIB
activin receptor type 2B
TGF-β superfamily
+ MUSCLE · AGING
PTH1R
GHSR
+12
2
cards
Cardiolipin
inner mitochondrial membrane
lipid target
+ AGING
PTH1R
IGF-1R
+10
2
cards
EPOR
erythropoietin receptor
type I cytokine receptor superfamily
+ CARDIOVASCULAR · INFLAMMATION
ACE
ANTIMICROBIAL
+14
2
cards
GDF-11
growth differentiation factor 11
TGF-β superfamily
+ MUSCLE · AGING
PTH1R
GHSR
+12
2
cards
OX2R
class A GPCR
+ WAKEFULNESS · AROUSAL · ENERGY-HOMEOSTASIS
1
cards
Actin (G-actin)
G-actin
cytoskeletal protein
+ MUSCLE
GHSR
IGF-1R
+6
1
cards
Anti-Aging
category
longevity
+ AGING · SKIN
PTH1R
IGF-1R
+13
1
cards
BRP-R
orphan-receptor ligand
+ WEIGHT LOSS · ANTI-OBESITY
GLP-1R
CCKAR
+7
1
cards
Fat Metabolism
category
1
cards
FSHR
FSH receptor
glycoprotein hormone receptor (class A GPCR)
+ REPRODUCTIVE
MC4R
GNRHR
+3
1
cards
GPR173
SREB3
rhodopsin-like GPCR (class A)
1
cards
KCNK2 / TREK-1
K2P (two-pore-domain) potassium channel family
1
cards
Mitochondrial
category
MDP
+ MUSCLE · AGING
PTH1R
GHSR
+12
1
cards
NPFFR2
Class A GPCR / RFamide receptor family
1
cards
NPY2R
Y2R
rhodopsin-like GPCR (class A)
1
cards
S1PR2
Class A GPCR / lysophospholipid receptor family
1
cards
SSTR2
+ ENDOCRINE
1
cards
UTS2R
urotensin II receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE
CALCR/RAMP
+6
0
cards
GH Secretagogue
GHRH
endocrine
+ MUSCLE · AGING
PTH1R
GHSR
+12