all targets

64 targets · sorted by activity
502 cards
ACE
angiotensin-converting enzyme
metalloprotease
+ CARDIOVASCULAR
CALCR/RAMP PTH1R +6
300 cards
Antimicrobial category
AMP
+ IMMUNE · INFLAMMATION
VPAC1 TACR1 +6
228 cards
GLP-1R
GLP-1 receptor
secretin receptor family (class B GPCR)
+ WEIGHT LOSS · DIABETES · GUT
NTSR1 CCKAR +14
199 cards
Anticancer category
+ CANCER
GNRHR IGF-1R
33 cards
OPRM1
mu-opioid receptor
rhodopsin-like GPCR (class A)
+ PAIN
CALCR/RAMP TACR1 +4
best 4
31 cards
CALCR/RAMP
calcitonin receptor
secretin receptor family (class B GPCR)
+ PAIN · CARDIOVASCULAR
ACE OPRM1 +12
29 cards
NTSR1
neurotensin-1 receptor
rhodopsin-like GPCR (class A)
+ BRAIN · GUT
GLP-1R CCKAR +17
26 cards
CCKAR
CCK1 receptor
rhodopsin-like GPCR (class A)
+ GUT · WEIGHT LOSS
GLP-1R NTSR1 +13
26 cards
VPAC1
VIP receptor 1
secretin receptor family (class B GPCR)
+ BRAIN · INFLAMMATION · GUT
ANTIMICROBIAL GLP-1R +22
25 cards
PTH1R
PTH receptor type 1
secretin-like GPCR (class B)
+ CARDIOVASCULAR · AGING
ACE CALCR/RAMP +18
23 cards
GCGR
glucagon receptor
secretin receptor family (class B GPCR)
+ WEIGHT LOSS · DIABETES
GLP-1R CCKAR +8
22 cards
MC3R
melanocortin-3 receptor
rhodopsin-like GPCR (class A)
+ WEIGHT LOSS · BRAIN
GLP-1R NTSR1 +18
20 cards
GHSR
ghrelin receptor
rhodopsin-like GPCR (class A)
+ MUSCLE · GUT · SLEEP
GLP-1R NTSR1 +14
19 cards
EDNRA
ETA receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE CALCR/RAMP +6
19 cards
TACR1
NK1 receptor
rhodopsin-like GPCR (class A)
+ PAIN · BRAIN · INFLAMMATION
ANTIMICROBIAL OPRM1 +20
18 cards
OPRD1
delta-opioid receptor
rhodopsin-like GPCR (class A)
+ PAIN · BRAIN
OPRM1 CALCR/RAMP +15
17 cards
GALR1
galanin-1 receptor
rhodopsin-like GPCR (class A)
+ BRAIN · GUT · WEIGHT LOSS
GLP-1R NTSR1 +21
17 cards
MC2R
melanocortin-2 receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE CALCR/RAMP +6
17 cards
MC4R
melanocortin-4 receptor
rhodopsin-like GPCR (class A)
+ WEIGHT LOSS · REPRODUCTIVE · BRAIN
GLP-1R NTSR1 +21
16 cards
CRHR2
CRF2 receptor
secretin-like GPCR (class B)
+ BRAIN · WEIGHT LOSS
GLP-1R NTSR1 +18
14 cards
GIPR
GIP receptor
secretin receptor family (class B GPCR)
+ WEIGHT LOSS · DIABETES
GLP-1R CCKAR +8
13 cards
ADCYAP1R1 / PAC1R
PAC1 receptor
secretin-like GPCR (class B)
+ PAIN · BRAIN · INFLAMMATION
ANTIMICROBIAL OPRM1 +20
12 cards
GnRHR
GnRH receptor
rhodopsin-like (class A GPCR)
+ CANCER · REPRODUCTIVE
ANTICANCER MC4R +5
12 cards
NPBWR1
neuropeptide B receptor 1
rhodopsin-like GPCR (class A)
+ BRAIN · PAIN
OPRM1 CALCR/RAMP +15
11 cards
GLP-2R
glucagon-like peptide 2 receptor
secretin-like GPCR (class B)
+ GUT
GLP-1R NTSR1 +6
10 cards
TACR2
NK2 receptor
rhodopsin-like GPCR (class A)
+ PAIN · GUT · INFLAMMATION
ANTIMICROBIAL GLP-1R +17
8 cards
KISS1R
kisspeptin receptor
rhodopsin-like GPCR (class A)
+ REPRODUCTIVE · BRAIN
NTSR1 VPAC1 +15
8 cards
Neuroprotective category
nootropic
+ BRAIN
NTSR1 VPAC1 +12
8 cards
OXTR
oxytocin receptor
rhodopsin-like GPCR (class A)
+ BRAIN · REPRODUCTIVE
NTSR1 VPAC1 +15
7 cards
AVPR1A
V1a receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE CALCR/RAMP +6
7 cards
IGF-1R
insulin-like growth factor 1 receptor
receptor tyrosine kinase
+ MUSCLE · CANCER · AGING
ANTICANCER PTH1R +14
7 cards
Longevity category
+ AGING
PTH1R IGF-1R +10
6 cards
AVPR2
vasopressin V2 receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE CALCR/RAMP +6
6 cards
Cosmeceutical category
+ SKIN
MC1R SKIN PEPTIDES +1
6 cards
SCTR
secretin receptor
secretin-like GPCR (class B)
+ GUT · BRAIN
GLP-1R NTSR1 +17
5 cards
AVPR1B
V1b receptor
rhodopsin-like GPCR (class A)
+ BRAIN
NTSR1 VPAC1 +12
5 cards
LHCGR
LH receptor
glycoprotein hormone receptor (class A GPCR)
+ REPRODUCTIVE
MC4R GNRHR +3
5 cards
Tissue Repair category
wound healing
+ INFLAMMATION · AGING
ANTIMICROBIAL VPAC1 +17
4 cards
MC1R
melanocortin-1 receptor
rhodopsin-like GPCR (class A)
+ SKIN · INFLAMMATION
ANTIMICROBIAL VPAC1 +9
3 cards
Activin A
INHBA
TGF-β superfamily
+ MUSCLE · AGING · INFLAMMATION
ANTIMICROBIAL VPAC1 +19
3 cards
GDF-8
myostatin
TGF-β superfamily
+ MUSCLE · WEIGHT LOSS · AGING
GLP-1R CCKAR +21
best 0.742
3 cards
GHRHR
Class B GPCR / secretin receptor family
3 cards
Immune category
3 cards
INSR
insulin receptor
receptor tyrosine kinase
+ DIABETES · AGING
GLP-1R PTH1R +13
3 cards
Skin Peptides category
cosmeceutical
+ SKIN
COSMECEUTICAL MC1R +1
2 cards
ActRIIB
activin receptor type 2B
TGF-β superfamily
+ MUSCLE · AGING
PTH1R GHSR +12
2 cards
Cardiolipin
inner mitochondrial membrane
lipid target
+ AGING
PTH1R IGF-1R +10
2 cards
EPOR
erythropoietin receptor
type I cytokine receptor superfamily
+ CARDIOVASCULAR · INFLAMMATION
ACE ANTIMICROBIAL +14
2 cards
GDF-11
growth differentiation factor 11
TGF-β superfamily
+ MUSCLE · AGING
PTH1R GHSR +12
2 cards
OX2R
class A GPCR
+ WAKEFULNESS · AROUSAL · ENERGY-HOMEOSTASIS
1 cards
Actin (G-actin)
G-actin
cytoskeletal protein
+ MUSCLE
GHSR IGF-1R +6
1 cards
Anti-Aging category
longevity
+ AGING · SKIN
PTH1R IGF-1R +13
1 cards
BRP-R
orphan-receptor ligand
+ WEIGHT LOSS · ANTI-OBESITY
GLP-1R CCKAR +7
1 cards
Fat Metabolism category
1 cards
FSHR
FSH receptor
glycoprotein hormone receptor (class A GPCR)
+ REPRODUCTIVE
MC4R GNRHR +3
1 cards
GPR173
SREB3
rhodopsin-like GPCR (class A)
1 cards
KCNK2 / TREK-1
K2P (two-pore-domain) potassium channel family
1 cards
Mitochondrial category
MDP
+ MUSCLE · AGING
PTH1R GHSR +12
1 cards
NPFFR2
Class A GPCR / RFamide receptor family
1 cards
NPY2R
Y2R
rhodopsin-like GPCR (class A)
1 cards
S1PR2
Class A GPCR / lysophospholipid receptor family
1 cards
SSTR2
+ ENDOCRINE
1 cards
UTS2R
urotensin II receptor
rhodopsin-like GPCR (class A)
+ CARDIOVASCULAR
ACE CALCR/RAMP +6
0 cards
GH Secretagogue
GHRH
endocrine
+ MUSCLE · AGING
PTH1R GHSR +12