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PAIN targets
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Target Name *
Alternative Names
UniProt ID
(optional)
Effect Type
(pick 1–3)
brain
sleep
pain
cardiovascular
immune
gut
diabetes
weight loss
reproductive
muscle
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inflammation
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00
all
64
01
BRAIN
15
02
SLEEP
1
03
PAIN
7
04
CARDIOVASCULAR
9
05
IMMUNE
1
06
GUT
9
07
DIABETES
4
08
WEIGHT LOSS
10
09
REPRODUCTIVE
6
10
MUSCLE
9
11
SKIN
4
12
INFLAMMATION
9
13
CANCER
3
14
AGING
13
7 targets
·
sorted by activity
activity
a-z
33
cards
OPRM1
mu-opioid receptor
rhodopsin-like GPCR (class A)
+ PAIN
CALCR/RAMP
TACR1
+4
best
4
31
cards
CALCR/RAMP
calcitonin receptor
secretin receptor family (class B GPCR)
+ PAIN · CARDIOVASCULAR
ACE
OPRM1
+12
19
cards
TACR1
NK1 receptor
rhodopsin-like GPCR (class A)
+ PAIN · BRAIN · INFLAMMATION
ANTIMICROBIAL
OPRM1
+20
18
cards
OPRD1
delta-opioid receptor
rhodopsin-like GPCR (class A)
+ PAIN · BRAIN
OPRM1
CALCR/RAMP
+15
13
cards
ADCYAP1R1 / PAC1R
PAC1 receptor
secretin-like GPCR (class B)
+ PAIN · BRAIN · INFLAMMATION
ANTIMICROBIAL
OPRM1
+20
12
cards
NPBWR1
neuropeptide B receptor 1
rhodopsin-like GPCR (class A)
+ BRAIN · PAIN
OPRM1
CALCR/RAMP
+15
10
cards
TACR2
NK2 receptor
rhodopsin-like GPCR (class A)
+ PAIN · GUT · INFLAMMATION
ANTIMICROBIAL
GLP-1R
+17