pe
pep-10337 v1 CC-BY-SA-4.0

Brain-signaling peptide that activates galanin receptors (CHEMBL592413)

A synthetic 24-amino-acid peptide that binds and switches on galanin receptors in the brain and nervous system; used only as a lab research tool.

statusbioassayed targetGALR1 length24 aa refs5
EARLY ENTRY This candidate is newly indexed — supporting evidence is still being added. Have a paper or data point? Contribute below.
status 5 / 5
prediction metrics boltz-2 2.2.1
ipTM0.853
pTM0.894
avg pLDDT76.7
ranking score0.784
STRUCTURE · PEP-10337 × GALR1
ranking0.784
target interface 4.5Å peptide drag rotate · ctrl+scroll zoom · right-click pan
boltz-2 2.2.1 · mmCIF ↓ download
sequence24 aa
1510152024
GWTLNSAGYLLG PRHYINLTRQRY
details expand to inspect
full evidence table1 metrics
metricvaluetool
Ki 0.3 nM GPCRDB/ChEMBL
3-letter notation
Gly-Trp-Thr-Leu-Asn-Ser-Ala-Gly-Tyr-Leu-Leu-Gly-Pro-Arg-His-Tyr-Ile-Asn-Leu-Thr-Arg-Gln-Arg-Tyr
recipeboltz-2 2.2.1
parametervalue
modelboltz-2 2.2.1
weights
hardwarevast_v100_32gb
mlx version
python
random seed1
msa strategycolabfold_local
runtime
predicted by
predicted at2026-05-22
citationbibtex
peptidemodel (2026). Brain-signaling peptide that activates galanin receptors (CHEMBL592413) (pep-10337, v1). PeptideModel. https://peptidemodel.com/card/pep-10337
@peptide{pep10337,
  sequence = {GWTLNSAGYLLGPRHYINLTRQRY},
  target   = {galr1},
  author   = {peptidemodel},
  year     = {2026},
  status   = {bioassayed}
}
related peptides 5 by signal overlap
clinical trials 0 trials · checked 2026-05-22
0
no registered clinical trials as of 2026-05-22; we'll re-check periodically
references 5 papers
[1]
Galanin receptors as a potential target for neurological disease
Freimann, K. et al. Expert Opinion on Therapeutic Targets 2015
supporting
[2]
Galanin Receptors and Ligands
Webling, K. et al. Frontiers in Endocrinology 2012
supporting
[3] supporting
[5]
Cloning and Expression of the Human Galanin Receptor GalR2
Bloomquist, B. et al. Biochemical and Biophysical Research Communications 1998
supporting
discussion no comments
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